编号:200388
CAS号:2022956-62-1
三字母:Ac-DVal-DGln-DIle-DVal-DTyr-DLys-Arg-Arg-Arg-Arg-Arg-Arg-Arg-Arg-Arg-NH2
描 述:T肽是PHF6的一种高度神经毒性的细胞渗透性类似物,可用于研究人类免疫缺陷病毒(HIV)感染。T肽可以诱导Tau肽聚集,防止细胞免疫抑制,提高败血症小鼠的存活率,并抑制手术切除后残留肿瘤细胞的生长。
编号:418004
CAS号:2703745-48-4/147159-51-1
三字母:H2N-DPhe-Cys-Tyr-DTrp-Lys-Cys-Thr-NH2(Disulfide Bridge:Cys2-Cys6)
描 述:TT-232-TFA是一种生长抑素类似物,作为sst1/st4生长抑素受体的肽激动剂。TT-232-TFA抑制人结肠癌细胞系中酪氨酸激酶的活性。显示TT-232-TFA抑制胰腺肿瘤细胞系中的增殖并诱导细胞凋亡。
编号:437254
CAS号:1234510-46-3/1824712-70-0
三字母:H2N-Sar-Arg-Val-Tyr-Ile-His-Pro-DAla-OH
描 述:TRV120027 TFA,一种血管紧张素II受体1型(AT1R)的β-抑制蛋白1偏向激动剂,在阻断G蛋白信号传导的同时与β-抑制素结合。
编号:192124
CAS号:108437-87-2
三字母:Pyr-Gln-Arg-Leu-Gly-Asn-Gln-Trp-Ala-Val-Gly-DPhe-Leu-Met-NH2
描 述:This bombesin receptor antagonist interacts only with the bombesin receptor. Because of this specificity, (D-Phe¹²)-Bombesin may be useful for defining the role of bombesin in various physiological or pathological processes.
编号:110738
CAS号:108437-89-4
三字母:Pyr-Gln-Arg-Tyr-Gly-Asn-Gln-Trp-Ala-Val-Gly-DPhe-Leu-Met-NH2
描 述:This bombesin analog is a specific antagonist of the bombesin receptor.
编号:116124
CAS号:118476-85-0
三字母:H2N-Tyr-DArg-Phe-Lys-NH2
描 述:The most selective µ-agonist reported to date. DALDA (YrFK-amide) should be useful not only as a research tool in basic opioid pharmacology but also for studying specifically peripheral µ-receptor interactions. Its very polar character should
编号:154671
CAS号:75644-90-5
三字母:H2N-Tyr-DSer-Gly-Phe-Leu-Thr-OH
描 述:The hexapeptide DSLET exhibits a very high specificity for the δ-receptor.
编号:200026
CAS号:926-78-3
三字母:H2N-DAla-DAla-DAla-DAla-OH
描 述:Tetra-D-丙氨酸,来自 Ochrobactrum anthropi 的 D-氨基肽酶的底物。
编号:121901
CAS号:118476-87-2
三字母:H2N-Tyr-DAla-Phe-Phe-NH2
描 述:TAPP, a relatively lipophilic peptide, shows high µ-receptor affinity, excellent µ-selectivity, and seems to be able to cross the blood-brain barrier.
编号:167345
CAS号:91224-37-2
三字母:H2N-DArg-Pro-Lys-Pro-Gln-Gln-DTrp-Phe-DTrp-Leu-Leu-NH2
描 述:substance P 的类似物,是选择性的神经激肽-1 受体 (NK1 receptor) 的拮抗剂。Spantide I可减少感染角膜的1型细胞因子和增强2型细胞因子IL-10,从而显著减少角膜穿孔。