编号:436835
CAS号:201422-04-0
三字母:Myristicacid-Lys-Ala-Leu-Arg-Arg-Gln-Glu-Ala-Val-Asp-Ala-Leu-OH
描 述:Autocamtide-2-相关抑制肽,肉豆蔻酰化醋酸酯是一种CaM激酶II抑制剂,通过预处理阻断体内吗啡寻求行为的恢复。它是自清-2-相关抑制肽的增强细胞渗透性衍生物。
编号:565781
CAS号:1402453-15-9
三字母:Ac-Arg-Phe(4NO2)-Diethylamine
描 述:ATIC-IN-1 是一种靶向氨基咪唑甲酰胺核糖核苷酸转化酶/肌苷一磷酸环化水解酶 ( ATIC ) 二聚化的抑制剂,Ki 值为 685 nM。ATIC 二聚化对其氨基咪唑甲酰胺核糖核苷酸 (AICAR) 转化酶活性至关重要。ATIC-IN-1 通过降低细胞数量和细胞分裂率表现出抗肿瘤活性。
编号:147507
CAS号:1621169-52-5
三字母:H2N-Ala-Trp-Arg-Gln-Asn-Thr-Arg-Tyr-Ser-Arg-Ile-Glu-Ala-Ile-Lys-Ile-Gln-Ile-Leu-Ser-Lys-Leu-Arg-Leu-CONH2
描 述:ACE-031是活化素受体型IIB (ActRIIB)的可溶形式,同时也是肌生成抑制素(myostatin)的抑制剂,能通过结合肌肉生长抑制素和其他肌肉的负性调节因子来促进肌肉生长,可用于Duchenne型肌营养不良症(DMD)的相关研究。
编号:153684
CAS号:143313-51-3
三字母:Ac-Tyr-Val-Ala-Asp-CHO
描 述:Ac-YVAD-CHO is a potent, specific, reversible inhibitor of caspase-1 (ICE). It displayed a Ki of 0.2 ± 0.1 nM for recombinant human caspase-1.
编号:160342
CAS号:189275-71-6
三字母:Ac-Trp-Glu-His-Asp-CHO
描 述:Ac-WEHD-CHO, a very potent reversible inhibitor of caspase-1 (ICE). It bears the optimal tetrapeptide recognition motif for this enzyme. With a Ki of 56 pM it belongs to the most potent reversible, peptide-based inhibitors described for any protease. For
编号:127786
CAS号:285570-60-7
三字母:Ac-Asp-Glu-Val-Asp-CMK
描 述:Ac-DEVD-CMK是一种细胞可渗透的、不可逆的胱天蛋白酶-3以及胱天蛋白酶-6、-7、-8和-10的抑制剂。它通常在高达100μM的浓度下用于检测胱天蛋白酶-3依赖性细胞凋亡在生物系统中的作用。
编号:175416
CAS号:35115-60-7
三字母:Pyr-Trp-Pro-Arg-Pro-Gln-Ile-Pro-Pro-OH
描 述:A nonapeptide originally isolated from the venom of the Brazilian pit viper Bothrops jararaca. Teprotide inhibits angiotensin-converting enzyme (ACE) in vitro and in vivo.
编号:190051
CAS号:75539-79-6
三字母:Cbz-DPhe-Phe-Gly-OH
描 述:A high level of inhibition of virus replication was obtained with this peptide, which resembles a region of a viral polypeptide.