皮啡肽(Dermorphin)

编号：151077

CAS号：

三字母：H2N-Tyr-DArg-Phe-Sar-Tyr-Pro-Ser-CONH2

描 述：是 Dermorphin 的类似物。Dermorphin 为两栖类皮肤中发现的天然七肽，为阿片受体激动剂。

编号：147636

CAS号：77614-16-5

三字母：H2N-Tyr-DAla-Phe-Gly-Tyr-Pro-Ser-CONH2

描 述：在两栖类皮肤中发现的一种天然七肽 μ-阿片受体 (MOR) 激动剂。Dermorphin 可用于抑制神经痛。

编号：132653

CAS号：100304-60-7

三字母：H2N-Tyr-DArg-Phe-Gly-CONH2

描 述：YrFG-amide, which is more stable to enzymatic cleavage, is the most potent of the (D-Arg²)-dermorphin fragments. It produces significant antinociception in morphinetolerant mice.

编号：116124

CAS号：118476-85-0

三字母：H2N-Tyr-DArg-Phe-Lys-CONH2

描 述：The most selective µ-agonist reported to date. DALDA (YrFK-amide) should be useful not only as a research tool in basic opioid pharmacology but also for studying specifically peripheral µ-receptor interactions. Its very polar character should

编号：121901

CAS号：118476-87-2

三字母：H2N-Tyr-DAla-Phe-Phe-CONH2

描 述：TAPP, a relatively lipophilic peptide, shows high µ-receptor affinity, excellent µ-selectivity, and seems to be able to cross the blood-brain barrier.

编号：144820

CAS号：736992-21-5/1606994-55-1/1849610-71-4

三字母：H2N-DArg-Dmt-Lys-Phe-CONH2

描 述：SS-31肽是一种心磷脂过氧化物酶抑制剂和线粒体靶向肽。它可以改善左心室和线粒体功能。SS-31肽可减轻人小梁网状细胞中的线粒体功能障碍和氧化损伤。它可以防止iHTM和GTM（3）细胞受到H2O2诱导的持续氧化应激。治疗慢性心力衰竭和线粒体肌病的II期临床试验正在进行中。

编号：159078

CAS号：119975-64-3

三字母：H2N-Tyr-DMet-Phe-His-Leu-Met-Asp-CONH2

描 述：Deltorphin，一种首先从南美青蛙Phyllomedusa sauvagei的皮肤提取物中分离出的肽，对应于预测的前体吗啡肽七肽。

编号：143999

CAS号：90549-86-3

三字母：H2N-Tyr-DArg-Phe-Sar-OH

描 述：A proposed µ-opioid receptor selective tetrapeptide analog of dermorphin. It showed more potent and longer-lasting analgesic activities than morphine.

编号：165528

CAS号：142689-18-7

三字母：H2N-Tyr-DAla-Phe-Gly-Tyr-Pro-Lys-CONH2

描 述：(Lys⁷)-Dermorphin is a mu1 receptor agonist with 20-30 times stronger analgesic properties than morphine.

编号：196927

CAS号：

三字母：H2N-Tyr-DAla-Phe-Trp-Asn-CONH2

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