编号:451725
CAS号:58970-76-6/65391-42-6
三字母:3-(r)-amino-2-(s)-hydroxy-4-phenylbutanoyl-(s)-leucine
描 述:Bestatin hydrochloride是氨基肽酶N(APN/CD13)抑制剂,其IC50值为14.9±3.4μM。
编号:153684
CAS号:143313-51-3
三字母:Ac-Tyr-Val-Ala-Asp-CHO
描 述:Ac-YVAD-CHO is a potent, specific, reversible inhibitor of caspase-1 (ICE). It displayed a Ki of 0.2 ± 0.1 nM for recombinant human caspase-1.
编号:133579
CAS号:149231-65-2
三字母:Ac-Tyr-Val-Ala-Asp-AMC
描 述:Ac-YVAD-AMC is a fluorogenic substrate for caspase-1 (ICE). It displayed a Km of 8.5 ± 0.5 µM for recombinant human caspase-1.
编号:160342
CAS号:189275-71-6
三字母:Ac-Trp-Glu-His-Asp-CHO
描 述:Ac-WEHD-CHO, a very potent reversible inhibitor of caspase-1 (ICE). It bears the optimal tetrapeptide recognition motif for this enzyme. With a Ki of 56 pM it belongs to the most potent reversible, peptide-based inhibitors described for any protease. For
编号:181876
CAS号:219137-97-0
三字母:Ac-Val-Glu-Ile-Asp-AMC
描 述:Ac-VEID-AMC, specific fluorogenic substrate for caspase-6.
编号:193145
CAS号:189684-53-5
三字母:Ac-Val-Asp-Val-Ala-Asp-pNA
描 述:Ac-VDVAD-pNA是caspase-2 的显色底物多肽,序列中含有5个氨基酸,是caspase-2 的首选底物,Km值为53μM。