编号:158432
CAS号:192723-42-5
三字母:MCA-Pro-Leu-Ala-Gln-Ala-Val-Dap(Dnp)-Arg-Ser-Ser-Ser-Arg-NH2
描 述:Mca-PLAQAV-Dpa-RSSSR-酰胺,一种荧光(FRET)肽底物,用于肿瘤坏死因子(TNF)转换酶(TACE,ADAM-17内肽酶)。
编号:125482
CAS号:5156-22-9
三字母:H2N-Leu-Trp-OH
描 述:LW 是一种存在于发酵乳中的 ACE 抑制性二肽,IC₅₀ 6.6 μM。氨肽酶 W 的底物,Km 0.57 mM 和 kcat 6770 min⁻¹。
编号:186395
CAS号:
三字母:H2N-Lys-Ala-Arg-Val-Nle-Phe(4NO2)-Glu-Ala-Nle-NH2
描 述:HIV-1 和 HIV-2 蛋白酶的敏感显色底物。H-1048 裂解的动力学参数:vmax 0.88 µM sec⁻¹,µg⁻¹, Km 15 µM, kcat 4.9 sec⁻¹.
编号:145310
CAS号:73167-83-6
三字母:Benzoyl-Gly-Phe-Arg-OH
描 述:Hip-Phe-Arg用作血管紧张素I转换酶和二肽基羧肽酶的底物。
编号:121540
CAS号:592544-81-5
三字母:MCA-Gly-Ser-Pro-Ala-Phe-Leu-Ala-Lys(Dnp)-DArg-NH2
描 述:Highly sensitive and selective cathepsin E FRET substrate derived from the cleavage site sequence of human α2-macroglobulin (Km = 1.9 µM; kcat/Km = 10.2 µM⁻¹s⁻¹ for human erythrocyte cathepsin E). The substrate was resistent to
编号:131637
CAS号:67368-29-0
三字母:H2N-Met-Arg-Phe-Ala-OH
描 述:H-Met-Arg-Phe-Ala-OH是来自人类红细胞的二肽基肽酶III和snapalysin的底物。它已被证明是从大鼠大脑中分离的脑啡肽生成内肽酶的竞争性抑制剂。
编号:118589
CAS号:201332-32-3
三字母:H2N-Ala-Ala-Pro-Leu-pNA
描 述:Good substrate (Km = 2.96 nM, kcat = 23.9 s⁻¹) for musk melon protease, an enzyme that enzymatic properties are similar to those of cucumisin and that seems to be a useful protease for the food industries. AAPL-pNA is also cleaved by guinea pig chyma