皮啡肽(Dermorphin)

编号：147636

CAS号：77614-16-5

三字母：H2N-Tyr-DAla-Phe-Gly-Tyr-Pro-Ser-NH2

描 述：在两栖类皮肤中发现的一种天然七肽 μ-阿片受体 (MOR) 激动剂。Dermorphin 可用于抑制神经痛。

编号：132653

CAS号：100304-60-7

三字母：H2N-Tyr-DArg-Phe-Gly-NH2

描 述：YrFG-amide, which is more stable to enzymatic cleavage, is the most potent of the (D-Arg²)-dermorphin fragments. It produces significant antinociception in morphinetolerant mice.

编号：116124

CAS号：118476-85-0

三字母：H2N-Tyr-DArg-Phe-Lys-NH2

描 述：The most selective µ-agonist reported to date. DALDA (YrFK-amide) should be useful not only as a research tool in basic opioid pharmacology but also for studying specifically peripheral µ-receptor interactions. Its very polar character should

编号：121901

CAS号：118476-87-2

三字母：H2N-Tyr-DAla-Phe-Phe-NH2

描 述：TAPP, a relatively lipophilic peptide, shows high µ-receptor affinity, excellent µ-selectivity, and seems to be able to cross the blood-brain barrier.

编号：143999

CAS号：90549-86-3

三字母：H2N-Tyr-DArg-Phe-Sar-OH

描 述：A proposed µ-opioid receptor selective tetrapeptide analog of dermorphin. It showed more potent and longer-lasting analgesic activities than morphine.

编号：196927

CAS号：

三字母：H2N-Tyr-DAla-Phe-Trp-Asn-NH2

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